6,495,366 6,495,532 6,500,150 6,503,062 6,503,184 6,503,231 6,505,059 6,512,939 6,514,500 6,520,326 6,520,747 6,520,936 6,520,938 D471,352 6,527,716 6,530,900 6,537,268 6,544,193 6,544,229 6,551,276 6,554,798 6,554,800 6,555,986 6,558,320 6,558,343 6,558,345 6,558,351 6,560,471 6,562,001 6,564,105 6,565,509 6,565,531 6,565,534 6,565,535 6,565,885 6,571,128 6,572,586 6,577,899 6,579,690 6,585,644 6,585,695 6,586,401 6,589,229 6,589,936 6,591,876 6,593,295 6,595,202 6,595,756 6,595,956 6,604,908 6,607,509 6,608,101 6,610,288 6,611,707 6,613,026 6,613,038 6,616,627 6,617,450 6,622,732 6,629,954 6,632,215 6,635,049 6,635,743 6,641,533 6,641,562 6,642,015 6,645,175 6,648,821 6,651,656 6,652,493 6,652,510 6,653,283 6,656,148 6,656,158 6,656,159 6,659,948 6,659,982 6,660,509 6,663,359
12/2002 12/2002 12/2002 1/2003 1/2003 1/2003 1/2003 1/2003 2/2003 2/2003 2/2003 2/2003 2/2003 3/2003 3/2003 3/2003 3/2003 4/2003 4/2003 4/2003 4/2003 4/2003 4/2003 5/2003 5/2003 5/2003 5/2003 5/2003 5/2003 5/2003 5/2003 5/2003 5/2003 5/2003 5/2003 5/2003 6/2003 6/2003 6/2003 7/2003 7/2003 7/2003 7/2003 7/2003 7/2003 7/2003 7/2003 7/2003 7/2003 8/2003 8/2003 8/2003 8/2003 8/2003 9/2003 9/2003 9/2003 9/2003 9/2003 10/2003 10/2003 10/2003 10/2003 11/2003 11/2003 11/2003 11/2003 11/2003 11/2003 11/2003 11/2003 11/2003 12/2003 12/2003 12/2003 12/2003 12/2003 12/2003 12/2003
Briggs
Bathurst et al. Gross et al. Gray et al.
Ni et al. Prausnitz et al. Kollias et al. Colvin et al. Bridon et al. Mclvor et al. Gray et al. Mann Funderburk et al. Shetler et al. Eppstein
Daily et al. Gibson et al. Abreu
Danby et al. Mann et al. Mann et al. Nezhadian et al. Moberg Causey, III et al. Neftel et al. Houben et al. Steil et al. Heller et al. Lebel et al.
Say et al. Mori et al. Winters
Zaias et al. Tarara et al. Lebel et al. Woj cik
Lebel et al. Bonnecaze et al. Lebel et al. Adair et al. Thorn et al. Connelly et al. Thorn et al. Safabash Bridon et al.
Gray et al. Gross et al. Bryant et al. Bobroff et al. Ni et al.
Edge et al. Prausnitz et al. Palasis et al. Bonutti et al. Willis et al. Stocker et al. Constantz Heruth Lemelson Robinson et al. Ebner et al. Causey, III et al. Peterson Vachon et al. Kriesel et al. Lebel et al. Demers et al. Das
Lord et al. Moses et al. Das et al. Mahoney et al. Flaherty Lebel et al. Douglas et al. Herman et al. Gray
6,665,909 6,666,845 6,669,663 6,669,668 6,669,669 6,671,554 6,685,664 6,687,546 6,689,073 6,689,100 6,689,108 6,689,607 6,689,747 6,692,456 6,692,457 6,694,191 6,699,218 6,699,219 6,702,779 6,703,217 6,709,417 6,711,436 6,716,190 6,716,193 6,721,582 6,723,072 6,726,656 6,728,560 6,733,446 6,734,162 6,734,186 6,736,795 6,737,401 6,740,059 6,740,072 6,740,075 6,740,655 6,749,403 6,749,587 6,750,311 6,752,299 6,752,785 6,752,787 6,753,177 6,753,328 6,755,811 6,758,810 6,766,183 6,768,425 6,770,067 6,770,729 6,774,120 6,784,274 6,792,982 6,796,956 6,796,957 6,800,071 6,800,663 6,801,420 6,804,544 6,805,687 6,805,693 6,808,369 6,808,506 6,809,507 6,809,653 6,810,290 6,811,533 6,811,534 6,813,519 6,814,715 6,817,990 6,821,949 6,824,529 6,827,702 6,830,558 6,830,564 6,840,922 6,843,782
12/2003 12/2003 12/2003 12/2003 12/2003 12/2003 2/2004 2/2004 2/2004 2/2004 2/2004 2/2004 2/2004 2/2004 2/2004 2/2004 3/2004 3/2004 3/2004 3/2004 3/2004 3/2004 4/2004 4/2004 4/2004 4/2004 4/2004 4/2004 5/2004 5/2004 5/2004 5/2004 5/2004 5/2004 5/2004 5/2004 5/2004 6/2004 6/2004 6/2004 6/2004 6/2004 6/2004 6/2004 6/2004 6/2004 7/2004 7/2004 7/2004 8/2004 8/2004 8/2004 8/2004 9/2004 9/2004 9/2004 10/2004 10/2004 10/2004 10/2004 10/2004 10/2004 10/2004 10/2004 10/2004 10/2004 10/2004 11/2004 11/2004 11/2004 11/2004 11/2004 11/2004 11/2004 12/2004 12/2004 12/2004 1/2005 1/2005
Collins et al. Hooper et al. Thompson Kleeman et al. Flaherty et al. Gibson et al. Levin et al.
Lebel et al.
Quay
Connelly et al. Lavi et al.
Ni et al.
Filvaroff et al. Eppstein et al. Flaherty Starkweather et al. Flaherty et al. Emig et al. .................. .. 604/131 Connelly et al. Herman et al. Houle et al. Duhaylongsod Glines et al. Neftel
Trepagnier et al. Flaherty et al. Kamen et al. Kollias et al. Lebel et al.
Van Antwerp et al. Maw et al.
Michel
Kim et al. Flaherty Starkweather et al. Lebel et al. Magee et al. Bryant et al. Flaherty
Van Antwerp et al. Shetler et al.
Van Antwerp et al. Causey, III et al. Stocker et al. Wands et al. Constantz
Lebel et al.
Walsh et al. Flaherty et al. Lorenzen et al. Van Antwerp Ferber et al.
Van Antwerp et al. Lincoln et al. Hartlaub et al. Carpenter et al. McConnell et al. Asgarzadeh et al. Talbot et al.
Van Antwerp et al. Dextradeur et al. Gray et al.
Gray et al. Lastovich et al. Morgan et al. Mann et al.
Lebel et al.
Lebel et al. Bowman, IV et al. Lebel et al. Bonutti et al.
Yap et al.
Bridon et al. Gross et al.
Lebel et al. Flaherty et al. Gray
Nielsen et al. Gross et al.
![[graphic]](http://www.google.com.au/patents?id=S1P_AQAAEBAJ&ie=ISO-8859-1&output=text&pg=PA6&img=1&zoom=3&hl=en&q=&cds=1&sig=ACfU3U26Vcueh5ZsVm6iByF8UhWPFQjMXw&edge=0&edge=stretch&ci=127,127,733,3)
Page 6 6,849,718 B2 2/2005 Kaelin, Jr. et al. 2004/0002682 A1 1/2004 Kovelman et al. 6,849,719 B2 2/2005 Shi et al. 2004/0029784 A1 2/2004 Hathaway 6,902,544 B2 6/2005 Ludin et al. 2004/0064086 A1 4/2004 Gottlieb et al. 6,936,029 B2 8/2005 Mann et al. 2004/0064096 A1 4/2004 Flaherty et al. 6,939,324 B2 9/ 2005 Gonnelli et al. 2004/ 0064097 A1 4/2004 Peterson 6,960,184 B2 11/2005 Willis et al. 2004/0073161 A1 4/2004 Tachibana 6,979,316 B1 12/2005 Rubin et al. 2004/0077000 A1 4/2004 Stocker et al. 7,011,234 B2 3/2006 Stradella 2004/0085215 A1 5/2004 Moberg et al. 7,014,625 B2 3/2006 Bengtsson 2004/0091374 A1 5/2004 Gray 7,022,107 B1 4/2006 Christensen et al. 2004/0092873 A1 5/2004 Moberg 7,108,686 B2 9/2006 Burke et al. 2004/0092893 A1 5/2004 Haider et al. 7,150,409 B2 12/2006 Gonnelli et al. 2004/0094823 A1 5/2004 Matsuno 7,204,823 B2 4/2007 Estes et al. 2004/0115067 A1 6/2004 Rush et al. 7,214,221 B2 5/2007 Fentress et al. .......... .. 604/890.1 2004/0116905 A1 6/2004 Pedersen et al. 7,250,037 B2 7/2007 Shermer et al. 2004/0126372 A1 7/2004 Banerjee et al. 7,337,922 B2 3/2008 Rake et al. 2004/0126373 A1 7/2004 Banerjee et al. 7,367,968 B2 5/2008 Rosenberg et al. 2004/0133163 A1 7/2004 Schiffmann 7,481,792 B2 1/2009 Gonnelli et al. 2004/0143216 A1 7/2004 Douglas et al. 7,530,968 B2 5/2009 Gonnelli ..................... .. 604/132 2004/0143217 A1 7/2004 Michel 7,534,226 B2 5/2009 Mernoe et al. 2004/0143218 A1 7/2004 Das 7,678,079 B2 3/2010 Shermer et al. 2004/0153032 A1 8/2004 Garribotto et al. 7,914,499 B2 3/2011 Gonnelli et al. ............ .. 604/186 2004/0155079 A1 8/2004 Shetler et al. 2001/0005781 A1 6/2001 Bergens et al. 2004/0167464 A1 8/2004 Ireland et al. 2001/0010238 A1 8/2001 Bynum 2004/0167470 A1 8/2004 Emig et al. 2001/0016710 A1 8/2001 Nason et al. 2004/0176725 A1 9/2004 Stutz et al. 2001/0027287 A1 10/2001 Shmulewitz et al. 2004/0209801 A1 10/2004 Brand et al. 2001/0031944 A1 10/2001 Peterson et al. 2004/0220456 A1 11/2004 Eppstein 2001/0037083 A1 11/2001 Hartlaub et al. 2004/0220525 A1 11/2004 Willis et al. 2001/0053891 A1 12/2001 Ackley 2004/0225281 A1 11/2004 Lorenzen et al. 2001/0056259 A1 12/2001 Skinkle et al. 2004/0247445 A1 12/2004 Nelson et al. 2002/0004015 A1 1/2002 Carlisle et al. 2004/0249363 A1 12/2004 Burke et al. 2002/0019612 A1 2/2002 Watanable et al. 2004/0250382 A1 12/2004 Collins et al. 2002/0040208 A1 4/2002 Flaherty et al. 2004/0254525 A1 12/2004 Uber et al. 2002/ 0045867 A1 4/ 2002 Nielsen et al. 2004/ 0260234 A1 12/2004 Srinivasan et al. 2002/0055460 A1 5/2002 Coolidge et al. 2004/0266678 A1 12/2004 Beeley et al. 2002/0061838 A1 5/2002 Holmquist et al. 2004/0267201 A1 12/2004 Agerup 2002/0072733 A1 6/2002 Flaherty 2005/0008661 A1 1/2005 Fereira et al. 2002/0077599 A1 6/2002 Wojcik 2005/0024175 A1 2/2005 Gray et al. 2002/0091358 A1 7/2002 Klitrnose 2005/0033232 A1 2/2005 Kriesel 2002/0095124 A1 7/2002 Palasis et al. 2005/0054988 A1 3/2005 Rosenberg et al. 2002/0123716 A1 9/2002 VanDiver et al. 2005/0065472 A1 3/2005 Cindrich et al. 2002/0123740 A1 9/2002 Flaherty et al. 2005/0070875 A1 3/2005 Kulessa 2002/0128594 A1 9/2002 Das et al. 2005/0112188 A1 5/2005 Eliaz et al. 2002/0138049 A1 9/2002 Allen et al. 2005/0119618 A1 6/2005 Gonnelli 2002/0147131 A1 10/2002 Coolidge et al. 2005/0137530 A1 6/2005 Campbell et al. 2002/0151842 A1 10/2002 Gonnelli et al. 2005/0137578 A1 6/2005 Heruth et al. 2002/0151846 A1 10/2002 Christenson et al. 2005/0171477 A1 8/2005 Rubin et al. 2002/0156418 A1 10/2002 Gonnelli et al. 2005/0171512 A1 8/2005 Flaherty 2002/0156464 A1 10/2002 Blischak et al. 2005/0177109 A1 8/2005 Azzolini 2002/0177809 A1 11/2002 Kriesel et al. 2005/0215850 A1 9/2005 Klein et al. 2002/0183693 A1 12/2002 Peterson et al. 2005/0234428 A1 10/2005 Spohn et al. 2002/0188259 A1 12/2002 Hickle et al. 2005/0245904 A1 11/2005 Estes et al. 2002/0198493 A1 12/2002 Diaz et al. 2005/0273083 A1 12/2005 Lebel et al. 2002/0198494 A1 12/2002 Diaz et al. 2005/0277912 A1 12/2005 John 2003/0009133 A1 1/2003 Ramey 2005/0278073 A1 12/2005 Roth 2003/0022823 A1 1/2003 Efendic 2006/0030838 A1 2/2006 Gonnelli 2003/0024508 A1 2/2003 Hellar et al. 2006/0069382 A1 3/2006 Pedersen 2003/0050237 A1 3/2003 Kim et al. 2006/0079862 A1 4/2006 Genosar 2003/0050623 A1 3/2003 Lord et al. 2006/0100578 A1 5/2006 Lieberman 2003/0073626 A1 4/2003 Hathaway et al. 2006/0122628 A1 6/2006 Solar et al. 2003/0100888 A1 5/2003 Spinello 2006/0150747 A1 7/2006 Mallett 2003/0125669 A1 7/2003 Safabash et al. 2006/0184119 A1 8/2006 Remde et al. 2003/0130619 A1 7/2003 Safabash et al. 2006/0184154 A1 8/2006 Moberg et al. 2003/0130647 A1 7/2003 Gray et al. 2006/0189939 A1 8/2006 Gonnelli et al. 2003/0135158 A1 7/2003 Gonnelli 2006/0200112 A1 9/2006 Paul 2003/0135160 A1 7/2003 Gray et al. 2006/0264831 A1 11/2006 Skwarek et al. 2003/0158520 A1 8/2003 Safabash et al. 2006/0264835 A1 11/2006 Nielsen et al. 2003/0163223 A1 8/2003 Blomquist 2007/0016170 A1 1/2007 Kovelman 2003/0167039 A1 9/2003 Moberg 2007/0060894 A1 3/2007 Dai et al. 2003/0195157 A1 10/2003 Natarajan et al. 2007/0073236 A1 3/2007 Mernoe et al. 2003/0199445 A1 10/2003 Knudsen et al. 2007/0088268 A1 4/2007 Edwards 2003/0199823 A1 10/2003 Bobroff et al. 2007/0100283 A1 5/2007 Causey, III et al. 2003/0212000 A1 11/2003 Van Antwerp 2007/0149925 A1* 6/2007 Edwards et al. ............ .. 604/141 2003/0216684 A1 11/2003 Fentress et al. ............... .. 604/81 2007/0167912 A1 7/2007 Causey et al. 2003/0216714 A1 11/2003 Gill 2007/0173761 A1 7/2007 Kanderian, Jr. et al. 2003/0220610 A1 11/2003 Lastovich et al. 2007/0179444 A1 8/2007 Causey et al. 2003/0225373 A1 12/2003 Bobroff et al. 2007/0239114 A1 10/2007 Edwards et al. 2003/0229309 A1 12/2003 Babkes et al. 2007/0287958 A1 12/2007 McKenzie et al. 2003/0233069 A1 12/2003 Gillespie et al. 2007/0287985 A1 12/2007 Estes et al.
![[graphic]](http://www.google.com.au/patents?id=S1P_AQAAEBAJ&ie=ISO-8859-1&output=text&pg=PA7&img=1&zoom=3&hl=en&q=&cds=1&sig=ACfU3U2eaCB2FJn3C_gFp2FqeGnCu6rP9A&edge=0&edge=stretch&ci=127,126,733,4)
Page 7 2008/0058719 A1 3/2008 Edwards et a1. WO 2008036509 A3 3/2008 2008/0091176 A1 4/2008 Alessi et a1. WO 2008139458 A3 11/2008 2008/0106431 A1 5/2008 Blomquist WO 2009013735 A1 1/2009 2008/0125701 A1 5/2008 Moberg et a1. WO 2009016637 A2 2/2009 2008/0139910 A1 6/2008 Mastrototaro et al. WO 2009081403 A2 7/2009 2008/0183060 A1 7/2008 Steil et a1. WO 2009125398 A2 10/2009 2008/0215006 A1 9/2008 Thorkild 2008/ 0249468 A1 10/2008 Edwards et a1. OTHER PUBLICATIONS 2008/0306436 A1 12/2008 Edwards et a1. _ _ _ 2008/0312512 A1 12/2008 BI-ukalo et a1‘ Capaldi, Treatments and devices for future diabetes management. 2008/0319383 A1 12/2008 Byland et a1. Nurs Times. 101(18): 30-32, 2005. 2009/ 0054867 A1 2/2009 Gravesen et al. Choi et al., Control of blood glucose by novel GLP-1 delivery using 2009/0062747 A1 3/2009 Saul biodegradable triblock copolyrner of PLGA-PEG-PLGA in type 2 58838822232 2} 3/588; garter t 1 diabetic rats. Pharm RCS. 21(5); 827-31, 2004. amSea' D ah al.I '1 GLP-1 d h -b 1 2009/0093772 A1 4/2009 Genosar et 31, ,,,,,,,,,,,,, ,, 604/246 on ey e.t ’ ntraVentncu.ar . re uces S on ut n0.t Ong term food mtake or body weight in lean and obese rats. Brain Res. 2009/0182277 A1 7/2009 Carter 779 1 2 t 75 83 1998 2009/0202608 A1 8/2009 Alessi 61211. (k' )' ' 1 1 ' f 1 1.k .d b d h 2009/0220358 A1 9/2009 Krivsky et 31‘ Druc er, Deve opr-nento g ucagon-1 epeptr e-1- ase p armaceu2009/0240232 A1 9/2009 Gonnelli et al‘ trcals as t11erapeut1c agents for the treatment of diabetes. Curr Pharm 2009/0247982 A1 10/2009 Kr616vi16h 61211. D93 704): 1399-412, 200l~ 2009/0281528 Al ll/2009 Grovender et al. Gappa et al., The effect of zinc-crystalized glucagon-like peptide-1 on insulin secretion of macroenca sulated ancreratic islets. Tissue FOREIGN PATENT DOCUMENTS Eng, 7(1), 3544, 2001, P P DE 36 34 7 2 5 4/ 1 988 Haak, New developments int he treatemnt of type 1 diabetes mellitus. DE 3634725 A1 4/1988 Exp Cin Endocrinol Diabetes, 107 Suppl 3: S108-13, 1999. DE 37 39 657 5/1988 Holst et al., On the treatment of diabetes mellitus with glucagon-like DE 3739657 A1 5/1988 peptid-1. Ann NY Acad Sci. 865:336-43, 1998. EP 0209677 A1 1/1987 Hui et al., The short half-life of glucagon-like peptide-1 in plasma EP 0401179 A1 l2;l990 does not reflect its long-lasting beneficial effects. Eur J Endocrinol. 513 8353252 :3 111221 1466 . . . . Joseph et al. Oral delivery of glucagon-l1ke pept1de-1 in a modrfied EP 0638324 A1 2/1995 . . . . . . EP 0937475 A2 8/1999 polymer preparation normalizes basal glycaem1a in diabetic db/db Ep 0902696 B1 3/2002 mice. Diabetologia. 43(10): 1319-28, 2000. EP 1 173197 B 1 12/2004 Toft-Nielsen et al., Continuous subcutaneous infusion of glucagonEP 1 5 l 2410 Al 3/2005 like peptide 1 lowers plasma glucose and reduces appetite in type 2 EP 1210136 B1 1/2006 diabetic patients. Diabetes Care. 22(7): 1137-43, 1999. GB 2 054 381 2/1981 Wang et al., Glucagon-like peptide-1 can reverse the age-related iI\§’L A decline in glucose tolerance in rats. J Clin Invest. 99(12): 2883-89, 1997. RU 2248223 C2 3/2005 Gonnelli, Robert R. Barnett International Needle-Free Injection Sys$8 tems presentation materials, Mar. 25, 2004, BioValve Technologies, wo wo-97/28835 8/1997 II.‘°' (10 Pages)‘. . . . W0 9808871 A1 3/1998 Smgapore Written Opinion from Smgapore Pat. App. No. W0 9947161 Al 9/1999 2008070302-5 dated Jan. 6, 2010. W0 9948546 A 9/1999 International Search Report for PCT/US2007/65363 dated Sep. 18, W0 0066138 A2 11/2000 2008 WO 0066142 A2 11/2000 Office Action for U.S.App1.No. 12/295,173 dated Jan. 26, 2010. WO 0100223 A2 1/2001 International Search Report for PCT/US2005/023818 dated Nov. 18, W0 0187322 A2 11/2001 2005, WO 02085406 A1 10/2002 011166 A61i611 f0f U.S. Appl. N6. 11/175,990 dated NOV. 10, 2009. WO 03008023 A1 IZZOO3 USPTO Non-Final Rejection mailed Jun. 10, 2010 in connection with 68 8221222 :2 3/588% . .. . International Search Report and Written Opinion marled Dec. 10, WO 03080160 A1 10/2003 . . . . . . WO 2004037195 A2 5/2004 2010 in connection w1t11 International Application No. PCT/US10/ wo 2004089335 A2 10/2004 52352 WO 2004094823 A2 11/2004 English Translation of First Office Action issued in connection with WO 2005046716 Al 5/2005 Chinese Application No: 200780020245.9, Dated Dec. 27, 2010. WO 2005048952 A2 6/2005 First EPO Examination Report issued in connection with European WO 2005060986 A1 7/2005 Application No. 01988242.2, Dated Dec. 27, 2010. WO 2007051139 A2 5/2007 WO 2007129317 A1 11/2007 * cited by examiner
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