DE60225701D1 - Ophthalmische depot-formulierungen zur periokkularen oder subkonjunktivalen verabreichung - Google Patents

Ophthalmische depot-formulierungen zur periokkularen oder subkonjunktivalen verabreichung

Info

Publication number
DE60225701D1
DE60225701D1 DE60225701T DE60225701T DE60225701D1 DE 60225701 D1 DE60225701 D1 DE 60225701D1 DE 60225701 T DE60225701 T DE 60225701T DE 60225701 T DE60225701 T DE 60225701T DE 60225701 D1 DE60225701 D1 DE 60225701D1
Authority
DE
Germany
Prior art keywords
periocular
depot formulations
subconjunctival administration
ophthalmic depot
ophthalmic
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
DE60225701T
Other languages
English (en)
Other versions
DE60225701T2 (de
Inventor
Markus Ahlheim
Michael Ausborn
David Bodmer
Christian Schoch
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Novartis AG
Original Assignee
Novartis AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis AG filed Critical Novartis AG
Publication of DE60225701D1 publication Critical patent/DE60225701D1/de
Application granted granted Critical
Publication of DE60225701T2 publication Critical patent/DE60225701T2/de
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0048Eye, e.g. artificial tears
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0048Eye, e.g. artificial tears
    • A61K9/0051Ocular inserts, ocular implants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605Excipients; Inactive ingredients
    • A61K9/1629Organic macromolecular compounds
    • A61K9/1641Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, poloxamers
    • A61K9/1647Polyesters, e.g. poly(lactide-co-glycolide)
DE60225701T 2001-09-14 2002-09-13 Ophthalmische depot-formulierungen zur periokkularen oder subkonjunktivalen verabreichung Expired - Lifetime DE60225701T2 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GBGB0122318.9A GB0122318D0 (en) 2001-09-14 2001-09-14 Organic compounds
GB0122318 2001-09-14
PCT/EP2002/010314 WO2003024420A1 (en) 2001-09-14 2002-09-13 Ophthalmic depot formulations for periocular or subconjunctival administration

Publications (2)

Publication Number Publication Date
DE60225701D1 true DE60225701D1 (de) 2008-04-30
DE60225701T2 DE60225701T2 (de) 2009-04-30

Family

ID=9922147

Family Applications (1)

Application Number Title Priority Date Filing Date
DE60225701T Expired - Lifetime DE60225701T2 (de) 2001-09-14 2002-09-13 Ophthalmische depot-formulierungen zur periokkularen oder subkonjunktivalen verabreichung

Country Status (25)

Country Link
US (4) US20040234611A1 (de)
EP (1) EP1429725B1 (de)
JP (3) JP2005504797A (de)
KR (1) KR20040030869A (de)
CN (2) CN1538835A (de)
AT (1) ATE389385T1 (de)
AU (1) AU2002342694B2 (de)
BR (1) BR0212475A (de)
CA (1) CA2455680C (de)
CO (1) CO5560548A2 (de)
DE (1) DE60225701T2 (de)
EC (1) ECSP044967A (de)
ES (1) ES2302849T3 (de)
GB (1) GB0122318D0 (de)
HK (1) HK1066733A1 (de)
HU (1) HU229453B1 (de)
IL (2) IL160027A0 (de)
MX (1) MXPA04002421A (de)
NO (1) NO333825B1 (de)
NZ (1) NZ531481A (de)
PL (1) PL203949B1 (de)
PT (1) PT1429725E (de)
RU (1) RU2316315C2 (de)
WO (1) WO2003024420A1 (de)
ZA (1) ZA200400524B (de)

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Also Published As

Publication number Publication date
IL160027A (en) 2009-11-18
JP2005504797A (ja) 2005-02-17
EP1429725A1 (de) 2004-06-23
RU2316315C2 (ru) 2008-02-10
EP1429725B1 (de) 2008-03-19
AU2002342694B2 (en) 2006-08-24
US20040234611A1 (en) 2004-11-25
ATE389385T1 (de) 2008-04-15
US20130122064A1 (en) 2013-05-16
JP2011026338A (ja) 2011-02-10
ES2302849T3 (es) 2008-08-01
ZA200400524B (en) 2004-11-17
PL203949B1 (pl) 2009-11-30
MXPA04002421A (es) 2004-05-31
CN1538835A (zh) 2004-10-20
NO333825B1 (no) 2013-09-23
DE60225701T2 (de) 2009-04-30
CA2455680A1 (en) 2003-03-27
ECSP044967A (es) 2004-03-23
NO20040917L (no) 2004-03-02
CA2455680C (en) 2010-07-20
BR0212475A (pt) 2004-08-24
US20120269894A1 (en) 2012-10-25
IL160027A0 (en) 2004-06-20
HUP0401568A3 (en) 2008-04-28
HK1066733A1 (en) 2005-04-01
PL368128A1 (en) 2005-03-21
CO5560548A2 (es) 2005-09-30
CN102008428A (zh) 2011-04-13
RU2004111596A (ru) 2005-04-20
US20080305172A1 (en) 2008-12-11
HUP0401568A2 (hu) 2004-11-29
GB0122318D0 (en) 2001-11-07
HU229453B1 (en) 2013-12-30
KR20040030869A (ko) 2004-04-09
WO2003024420A1 (en) 2003-03-27
JP2013147516A (ja) 2013-08-01
NZ531481A (en) 2005-12-23
PT1429725E (pt) 2008-06-18

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